Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ InSolution™ Tetrahydrouridine
Tetrahydrouridine is a potent competitive inhibitor of cytidine deaminase.
MilliporeSigma™ Calbiochem™ Camptothecin, Camptotheca acuminata
A cell-permeable DNA topoisomerase I inhibitor.
MilliporeSigma™ Calbiochem™ Casein Kinase II Inhibitor III, TBCA
The Casein Kinase II Inhibitor III, TBCA, also referenced under CAS 934358-00-6, controls the biological activity of Casein Kinase II. This small molecule/inhibitor is primarily used for Phosphorylation and Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Collagenase Inhibitor I
The Collagenase Inhibitor I controls the biological activity of Collagenase. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ Adenosine Receptor Agonist, NECA
A cell-permeable adenosine analog that acts a potent non-selective agonist of adenosine receptors (Ki = 14 nM, 20 nM
MilliporeSigma™ Calbiochem™ Focal Adhesion Kinase Inhibitor III
A cell-permeable pyrazolobenzothiazinedioxide compound that targets and locks FAK in its inactive conformation, resulting in preincubation time-dependent inhibition in kinase assays and FAK autophosphorylation in human prostate cancer PC3M-luc cells (IC50
MilliporeSigma™ Calbiochem™ 1-Pyrrolidinecarbodithioic Acid, Ammonium Salt
Cell permeable. Inhibits the induction of NOS activity in rat alveolar macrophages. Prevents apoptosis in human HL-60 cells and thymocytes, but induces apoptosis in human and rat smooth muscle cells.
MilliporeSigma™ Calbiochem™ mGluR5 Antagonist, MTEP
The mGluR5 Antagonist, MTEP, also referenced under CAS 329205-68-7, controls the biological activity of mGluR5. This small molecule/inhibitor is primarily used for Neuroscience applications.
MilliporeSigma™ Calbiochem™ 2-Chloro-2'-deoxyadenosine
A deoxyadenosine analog that displays strong antileukemic and immunosuppressive activity.
MilliporeSigma™ Calbiochem™ Meloxicam
A cell-permeable, non-steroidal anti-inflammatory drug (NSAID) of the oxicam family which preferentially inhibits the inducible isoform of COX-2 (IC50 = 4.7 μM) relative to COX-1 (IC50 = 36.6 μM).
MilliporeSigma™ Calbiochem™ α-Naphthyl Acid Phosphate, Monosodium Salt
α-Naphthyl Acid Phosphate, Monosodium Salt - CAS 81012-89-7, is a broad-spectrum protein phosphatase inhibitor.
MilliporeSigma™ Calbiochem™ PTP CD45 Inhibitor
The PTP CD45 Inhibitor, also referenced under CAS 345630-40-2, controls the biological activity of PTP CD45. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Pifithrin-α
A cell-permeable chemical inhibitor of p53.
MilliporeSigma™ Calbiochem™ InSolution™ Casein Kinase I Inhibitor, D4476
The InSolution™ Casein Kinase I Inhibitor, D4476 controls the biological activity of Casein Kinase I. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ ACA
A cell-permeable inhibitor of phospholipase A2 that blocks epinephrine-stimulated thromboxane production in platelets.